P-gp
P-gp (P-glycoprotein) is a ATP-binding cassette transproters which overepxressed in multidrug-resistance cancer cells. It functions in pumping drug out of cell and lower intracellular drug concentration.
- C3840 Estradiol 17-(β-D-Glucuronide) (sodium salt)Summary: 多药耐药蛋白2(MRP2)的底物
- C3897 Estradiol 3-(β-D-Glucuronide) (sodium salt)Summary: 多药耐药蛋白2(MRP2)的底物
- C3610 HypophyllanthinSummary: P-糖蛋白(P-gp)抑制剂
- C3140 Rhodamine 123 (chloride)中文名: 罗丹明123Summary: 膜可渗透的阳离子染料,用作流出泵P-糖蛋白的底物
- B1167 Dofequidar fumarateSummary: MDR逆转剂
- A8549 LY335979 (Zosuquidar 3HCL)1 Citation中文名: 唑喹达三盐酸盐Target: P-glycoprotein (P-gp)Summary: Pgb(P糖蛋白)抑制剂
- A3956 ZosuquidarTarget: P-glycoprotein (P-gp)|Cytochrome P450 (CYP450)Summary: MDR调节剂
- A3859 Tariquidar methanesulfonate, hydrate中文名: 他立喹达二甲磺酸盐六水合物Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂
- A8208 Tariquidar2 Citation中文名: 他立喹达Target: P-glycoprotein (P-gp)Summary: P-糖蛋白抑制剂